opioid receptor การใช้

• "Naltrexone simply blocks the opioid receptors so the endorphines can't get there.
• Menthol's analgesic properties are mediated through a selective activation of ?-opioid receptors.
• These endorphins likely operate on the same opioid receptors that naloxone blocks.
• Levorphanol is 6-8 times as potent as morphine at the mu-opioid receptor.
• Eletriptan has no significant affinity or pharmacological activity at muscarinic; or opioid receptors.
• Descending pathways also activate opioid receptor-containing parts of the spinal cord.
• This points to a role for opioid receptors in mating behaviors.
• More recent investigations, however, discovered opioid receptors on peripheral sensory neurons.
• In vertebrates, neuromodulators that moderate pain by interacting with opioid receptors.
• Loperamide is a ?-opioid receptor agonist that works in the intestines.
• Unlike most benzodiazepines, tifluadom has no activity at the ?-opioid receptor.
• 6'- GNTI is an extremely biased agonist of the ?-opioid receptor.
• Cyprodime is a selective opioid antagonist which blocks the ?-opioid receptors.
• Cyprenorphine has mixed agonist antagonist effects at opioid receptors, like those of buprenorphine.
• Additionally, opioid drugs suppress nociceptions by binding to endogenous opioid receptors.
• Inflammatory pain is also blunted by endogenous opioid peptides activating peripheral opioid receptors.
• The prototypical ?-opioid receptor agonist is morphine, the primary psychoactive alkaloid in opium.
• Three known kinds of opioid receptors have been identified : delta ( ? ).
• The four main opioid receptor types ( primitive jawless fishes.
• Kyotorphin has an analgesic effect, but it does not interact with the opioid receptors.